Xermelo Drug Interactions
Currently displaying a list of 352 drugs known to interact with Xermelo (telotristat).
- 28 major drug interactions
- 317 moderate drug interactions
- 7 minor drug interactions
Medications known to interact with Xermelo
Note: Showing generic names only.
A
- abemaciclib
- abiraterone
- acalabrutinib
- albendazole
- alfentanil
- aliskiren
- alpelisib
- alprazolam
- amiodarone
- amlodipine
- amprenavir
- apixaban
- apremilast
- aprepitant
- aprocitentan
- aripiprazole
- armodafinil
- asenapine
- astemizole
- atazanavir
- atogepant
- atorvastatin
- avacopan
- avanafil
- avapritinib
- axitinib
B
- bedaquiline
- belumosudil
- bepridil
- betamethasone
- bexarotene
- boceprevir
- bortezomib
- bosentan
- bosutinib
- brentuximab
- brexpiprazole
- brigatinib
- bromocriptine
- budesonide
- buprenorphine
- bupropion
- buspirone
- butorphanol
C
- cabazitaxel
- cabozantinib
- capivasertib
- capmatinib
- carbamazepine
- cariprazine
- ceritinib
- cerivastatin
- cevimeline
- chlorotrianisene
- cinacalcet
- cisapride
- citalopram
- clarithromycin
- clonazepam
- clorazepate
- cobimetinib
- codeine
- conjugated estrogens
- copanlisib
- cortisone
- crizotinib
- cyclosporine
D
- daclatasvir
- dapsone
- daridorexant
- darifenacin
- darolutamide
- darunavir
- dasatinib
- dehydroepiandrosterone
- delavirdine
- dexamethasone
- dihydroergotamine
- diltiazem
- disopyramide
- docetaxel
- donepezil
- doravirine
- doxorubicin
- doxorubicin liposomal
- dronedarone
- dutasteride
- duvelisib
E
- efavirenz
- elacestrant
- elagolix
- eletriptan
- eliglustat
- encorafenib
- enfortumab vedotin
- entrectinib
- enzalutamide
- eplerenone
- erdafitinib
- ergonovine
- ergotamine
- erlotinib
- erythromycin
- estazolam
- estradiol
- estrone
- estropipate
- eszopiclone
- ethinyl estradiol
- ethosuximide
- etonogestrel
- etoposide
- etravirine
- everolimus
- exemestane
F
- fedratinib
- felodipine
- fenfluramine
- fentanyl
- fesoterodine
- fexinidazole
- finerenone
- flibanserin
- fludrocortisone
- flurazepam
- fosamprenavir
- fosaprepitant
- fostamatinib
- fostemsavir
G
H
I
- ibrexafungerp
- idelalisib
- imatinib
- indinavir
- infigratinib
- irinotecan
- irinotecan liposomal
- isavuconazonium
- isotretinoin
- isradipine
- istradefylline
- itraconazole
- ivabradine
- ivacaftor
- ivermectin
- ixabepilone
- ixazomib
K
L
- lapatinib
- larotrectinib
- lazertinib
- lefamulin
- lemborexant
- lenacapavir
- leniolisib
- letrozole
- levamlodipine
- levobupivacaine
- levoketoconazole
- levomethadyl acetate
- levonorgestrel
- lidocaine
- linagliptin
- lonafarnib
- loratadine
- lorlatinib
- lovastatin
- lumateperone
- lurasidone
- lurbinectedin
M
- macimorelin
- macitentan
- maraviroc
- maribavir
- mavacamten
- medroxyprogesterone
- mefloquine
- megestrol
- methadone
- methylergonovine
- methylprednisolone
- methysergide maleate
- mibefradil
- midazolam
- mifepristone
- mirabegron
- mirtazapine
- mitapivat
- mobocertinib
- modafinil
N
- naldemedine
- naloxegol
- nefazodone
- nelfinavir
- nevirapine
- nicardipine
- nicotine
- nifedipine
- nilotinib
- nimodipine
- nintedanib
- nirogacestat
- nisoldipine
- nitisinone
- norethindrone
- norgestrel
O
- octreotide
- olaparib
- oliceridine
- olutasidenib
- omaveloxolone
- ondansetron
- osilodrostat
- osimertinib
- oxybutynin
- oxycodone
P
- paclitaxel
- paclitaxel protein-bound
- pacritinib
- palbociclib
- palovarotene
- panobinostat
- paricalcitol
- pazopanib
- pemigatinib
- perampanel
- pexidartinib
- pimavanserin
- pirtobrutinib
- pomalidomide
- ponatinib
- praziquantel
- prednisolone
- prednisone
- pretomanid
- progesterone
- propofol
Q
R
- ramelteon
- ranolazine
- red yeast rice
- relugolix
- repaglinide
- repotrectinib
- revumenib
- ribociclib
- rifabutin
- rilpivirine
- rimegepant
- ripretinib
- ritlecitinib
- ritonavir
- rivaroxaban
- roflumilast
- rolapitant
- romidepsin
- ruxolitinib
S
- saquinavir
- saxagliptin
- selegiline
- selpercatinib
- selumetinib
- sertraline
- sildenafil
- silodosin
- simvastatin
- sirolimus
- sirolimus protein-bound
- solifenacin
- sonidegib
- sorafenib
- sotorasib
- sparsentan
- stiripentol
- sufentanil
- sunitinib
- suvorexant
- suzetrigine
T
- tacrolimus
- tadalafil
- tamoxifen
- tamsulosin
- tasimelteon
- tazemetostat
- telaprevir
- telithromycin
- temsirolimus
- teniposide
- tepotinib
- terfenadine
- testosterone
- testosterone topical
- thiotepa
- tiagabine
- ticagrelor
- tinidazole
- tipranavir
- tofacitinib
- tolterodine
- tolvaptan
- toremifene
- trabectedin
- tramadol
- trazodone
- tretinoin
- triamcinolone
- triazolam
- troglitazone
- troleandomycin
- tucatinib
U
V
- valbenazine
- valdecoxib
- vandetanib
- vemurafenib
- venlafaxine
- verapamil
- vilazodone
- vinblastine
- vincristine
- vincristine liposome
- vinorelbine
- voclosporin
- vonoprazan
- vorapaxar
- voriconazole
Z
Xermelo alcohol/food interactions
There are 2 alcohol/food interactions with Xermelo (telotristat).
Xermelo disease interactions
There are 3 disease interactions with Xermelo (telotristat) which include:
More about Xermelo (telotristat)
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Related treatment guides
Drug Interaction Classification
Highly clinically significant. Avoid combinations; the risk of the interaction outweighs the benefit. | |
Moderately clinically significant. Usually avoid combinations; use it only under special circumstances. | |
Minimally clinically significant. Minimize risk; assess risk and consider an alternative drug, take steps to circumvent the interaction risk and/or institute a monitoring plan. | |
No interaction information available. |
Further information
Always consult your healthcare provider to ensure the information displayed on this page applies to your personal circumstances.